O. I. Panasenko, A. A. Safonov, T. O. Samura, I. V. Melnik, V. A. Salionov, A. S. Gotsulya, V. P. Buryak, N. A. Postol, R. A. Sherbina, A. A. Kremzer, I. M. Keitlyn, T.V. Panasenko

Zaporozhye State Medical University

 

COLLECTIONS FOR ANALYTICAL TOXICOLOGY.

TRANSPORT AND STORAGE

 

It is usually advisable to contact the laboratory by telephone in advance to discuss urgent or complicated cases. Most specimens, particularly blood and urine, may be sent by post if securely packaged in compliance with current regulations. However, if legal action is likely to be taken on the basic of the results, it is important to be able guarantee the identity and integrity of the specimen from when it is of the specimen from when it is collected through to the reporting of the result. Thus, such samples should be protected during transport by the use of tamper- evident seals and should, ideally, be submitted .In person to the laboratory by the coroner’s officer or other investigating personnel. Chain of custody is a term used to refer to the process used to maintain and document the history of the specimen (see BOX 1).

BOX 1. Chain of custody documents. Name of the individual collecting the specimen. Name of each person or entity subsequently having custody of it, and details of how it has been stored. Dates/times the specimen was collected or transferred. Specimen or postmortem number. Name of the subject or deceased. Brief description of the specimen. Record of the condition of tamper-evident seals.

Fully validated assays must include data on the stability of the analyte under specified storage conditions. In the absence of other information, biological specimens should be stored at 2-8 °C prior to analysis, if possible, and ideally any specimen remaining after the analysis should be kept at 2-8 °C for 3-4 weeks in case further analyses are required. In view of the medico legal implications of some poison cases (e.g. if it is not clear how the poison was administered or if the patient dies) then any specimen remaining should be kept (preferably at -20 °C) until investigation of the incident is concluded. With regard to drugs, some compounds such as clonazepam, cocaine, nifedipine, nitrazepame, thiol drugs, and many phenothiazines and their metabolites are unstable in biological samples at room temperature. Exposure to sunlight can cause up to 99% lass of clonazepam in serum after 1h at room temperature. Covering  the outside of the sample tube in aluminum foil is a simple precaution in such cases. N-Glucuronides such as nomifensine N-Glucuronide are unstable and may be present in plasma at high concentration: on decomposition the parent compound us reformed. Some compounds unstable in whole blood or plasma are listed in (Table 1).

Solid sodium fluoride (2%, w/v) may be added to inhibit microbial and some other derivative enzymes. Esters (including carbonates and organophosphates) may be rapidly. Hydrolyzed by plasma esterase’s, including cholinesterase. If physostigmine or cocaine is to be measured accurately, the blood should be drawn into tubes containing an excess of neostigmine. Storage at -20 °C or below is recommended if the analysis cannot be performed immediately and if the stability of the analyte is unknown. However, even this may not be ideal because N-and S-oxyde may be reduced to the parent compounds.

Table 1

Some drugs, metabolites and other poisons unstable in whole blood or plasma

Volatile Compound(s)

No-volatile Compound(s)

Aerosol propellants, anesthetic gases, carbon monoxide, ethanol, chlorvynyl, hydrogen cyanide, mercury, methanol, nicotine, OP nerve agents, organic solvents, paraldehyde, volatile nitrites (amyl nitrite, etc.).

Acyl glucuronide metabolites, amiodarone, bupropion, carbonate esters, esters (aspirin, benzocaine, cocaine), gluceryl trinitrate, N-glucuronide metabolites, insulin, lysergic acid diethylamide, nitrobenzodiazepines, nitrophenyl-pyridines, olanzapine, N-oxide metabolites, S-oxide metabolites, paracetamole, peroxides, phenelzine, rifampicin, sirolimus, thalidomide, thiopental, zopiclone.

Quinols such as 4-hydroxypranolol and some sulfur-containing compounds such as olanzapine, on the other hand, are readily oxidized and stabilization b addition of a reducing agent such as ascorbate or sodium metabisulfite is necessary, but in the case of olanzapine, for example, there is the possibility of reducing the N-oxide by such an addition. Hydrolyzed by plasma esterase’s, including cholinesterase. If physostigmine or cocaine is to be measured accurately, the blood should be drawn into tubes containing an excess of neostigmine. Storage at -20 °C or below is recommended if the analysis cannot be performed immediately and if the stability of the analyte is unknown. However, even this may not be ideal because N-and S-oxyde may be reduced to the parent compounds.

Quinols such as 4-hydroxypranolol and some sulfur-containing compounds such as olanzapine, on the other hand, are readily oxidized and stabilization b addition of a reducing agent such as ascorbate or sodium metabisulfite is necessary, but in the case of olanzapine, for example, there is the possibility of reducing the N-oxide by such an addition. Storage at -5 to -70 °C should b accompanied by basic precautions to accompanied by basic precautions to preserve sample integrity (see Box 2). The requirements of the local ethics committee and other guidance on the retention and storage of clinical samples must be complied with.

Box 2. Guidance on freezer storage of samples. Do not freeze whole blood if plasma or serum is not be analyzed. Ensure that labelling is waterproof. Ensure tubes are tightly sealed and well filled, but do not overfill tubes, especially glass tubes. Do not keep too long to minimize freeze-drying effects. Keep a record of freezer contents. Keep a continuous record of freezer temperature. Fit an alarm in case of freezer failure.

Plasticizers, particularly phthalates, may originate from plastic bags used to store transfusion  blood, infusion tubing, and from soft plastic closures for blood tulles. Such compounds are often retained on reversed phase HPLC systems and show good absorption at 254 nm and below. Polyvinylchloride (PVC), for example, can contain up to (40%, w/w) di-2-ethylhexyl phthalate and compound of up to about 0,5 gl-1 have been reported after storage of plasma in PVC bags for 14 days [1]. A further consideration is that postmortem specimens may contain putrefactive bases such as phenylethylamines and indole, which may interfere in the analysis of amfetamines and other stimulants. Hexenal may arise from breakdown of fatty acids. Gas chromatography retention data and mass spectra of a number of plasticizers, pollutants, and other substances that may be encountered in toxicological analyses have been reported [2]. Modern blood-collection tubes may contain a range of additives including surfactants, which may interfere in immunoassays, for example [4].

Drug may arise from unexpected sources including food and over-the-counted (OTC) medicines. Quinine may originate from ingestion of domestic water, from example, caffeine from caffeinated beverages (tea, coffee, cola) and some proprietary stimulants, chloraquine and related compounds from malaria prophylaxis, and pholcodine and other opiate analogues from cough and cold cures. Morphine is a constituent of some antidiarrheal preparations. A caffeine metabolite, paraxanthine, may be a problem in the PLC theophylline assays [3]. Lidocaine-contaiing gel is commonly is commonly used as a lubricant during procedures such as bladder catheterization or bronchoscopy, and measurable plasma concentrations of lidocaine and some metabolites may be attained.

The alkaloids emetine and cephalline, and their metabolites, have been detected in stomach contents, plasma, and in urine other syrup of ipecacuanna (ipecac) was given  to induce  vomiting, especially in children, although this form of treatment is no longer recommended practice. Sedative (CT) seams, lumbar puncture, or other investigations. Neuromuscular blocking agents such as atracurium, which is metabolized to laudanosine, and vecuronium, may be encountered in samples from patiens undergoing mechanical ventilation. 1.3-Propanediol (propylene glycol) is used us a vehicle in i. v. infusions. Benzoic acid, which is metabolized to hippuric acid, is used as a preservative in some drugs and foods. The antibiotic metronidazole is often encountered in samples from hospitalized patients. Iodinated hippuric acids are used as X-ray contrast media.

Alcohols may originate from skin cleansing swabs. Such compounds and drugs given in emergencies, anticonvulsants, for example, may not be recorded on record sheets. Some compounds or their metabolites may have very long plasma half-lives. Chlorpromazine metabolites, for example, have been reported in urine many months after stopping therapy. Contamination with trace elements is a particularly difficult area. Contamination with volatiles, such as solvents used in the laboratory, must be guarded against if one of the solvents in question is to be tested for in a biological or related sample. Glassware and other items must be kept clean and tested regularly for contamination uva internal quality control.

SUMMARY. Although not in the immediate control of the laboratory, every effort must be made to ensure appropriate priority is given to sample collection and handling because if this us not teepee properly all subsequent effort us wasted. Care in sample collection is especially important in postmortem and overt medico legal work, but even in clinical work effort in providing advance information to clinicians and pathologists on sample requirements (side of collection, volume, addition of sodium fluoride, etc.) and feedback on the problems that will arise when mistakes are made can only prove beneficial.

REFERENCES

1.   Dine T., Luyckx M., Cazin M., Brunet C., Cazin I. C, Goudaliez F. Rapid determination by high performance liquid chromatography of di-2-ethylhexyl phthalate in plasma stored in plastic bags // Biomed. Chromatogr., 1991. - Vol. 5. - P. 94 - 97.

2.   Pfleger K., Maurer H. H, Weller A. Mass Spectral and GC Data of Drugs, Pollutants. Pesticides and their Metabolites, 2007, 3rd edn, Wiley-VCH, Weinheim.

3.   Stankovic A. K., Parmar G. Assay interferences from blood collection tulles: a Cautionary note. ClinChem., 2006. - Vol. 52. - P. 1627 - 1628.

4.   Rowe D. I., Watson I. D., Williams I., Berry D. J. The clinical use and measurement of theophylline Ann. Clin. Biochem., 1988. - Vol. 25. - P. 4 - 26.