Zemlyanskaya N.A., Kolbasina L.P., Kushnir K.G., Lavrinovskaya O.M.

SI “Crimea State Medical University named after S. I. Georgievsky”

Human organism adaptation potential development in patients with chronic hypertonic disease in the conditions of health resort rehabilitation

 

Melatonin is also known chemically as N-acetyl-5-methoxytryptamine, is a naturally occurring compound found in animals, plants, and microbes. In animals, circulating levels of the hormone melatonin vary in a daily cycle, thereby allowing the entrainment of the circadian rhythms of several biological functions.

Many biological effects of melatonin are produced through activation of melatonin receptors, while others are due to its role as a pervasive and powerful antioxidant, with a particular role in the protection of nuclear and mitochondrial DNA.

Melatonin impact on cardiovascular system is manifested by decrease of systolic arterial pressure in rest and decrease of systolic pressure growth in case of psychoemotional test, which says about cardiovascular system limited stress reactivity. Influence of melatonin on cardiovascular system manifested by decrease of systolic blood pressure at rest within the physiological rationality and reduce increase of systolic blood pressure during the psycho-emotional test, that shows the restriction of stress reaction of cardiovascular system.

      On the basis of notions, that hypertonic disease (essential hypertension) in a certain sense is the disease of maladjustment, justified the study of melatonin production in this pathology.

Cardiac output and peripheral resistance are the two determinants of arterial pressure. and so blood pressure is normally dependent on the balance between cardiac output and peripheral resistance. Cardiac output is determined by stroke volume and heart rate; stroke volume is related to myocardial contractility and to the size of the vascular compartment. Peripheral resistance is determined by functional and anatomic changes in small arteries and arterioles. The pathophysiology of essential hypertension is an area of research, and until now remains not well understood, but many theories have been proposed to explain this.

If to say that hypertonic disease partially is the disease of disadaptation (essential hypertension) the studying of melatonin production in case of such pathology is justified. When patients with hypertonic disease have the rehabilitation in health resorts the fact of migration to new climatic zone and changes of common regimen may cause tension of adaptation processes and circadian deregulation. Regulatory systems tension and organism functional reserves mobilization is the “price” for adaptation in such conditions.

Certain researches shown that melatonin supplementation in the evening in premenopausal women produces an improvement in thyroid function and gonadotropin levels, as well as restoring fertility and menstruation and preventing the depression associated with the menopause. And as we know, in women hypertonic disease usually develops in this age.

  The purpose of our investigation is optimization the adaption period at the sanatorium rehabilitation of patients having hypertension by effects of melatonin on desynchronosis processes.  The determination and intensity of adaptation is measured by 6-hydroxymelatoninsulphate (6-HMS) excretion in nocturnal urine of patients with hypertonic disease in health resort conditions. Analyzing of adaptation potential is such patients before and after melatonin drug intake.   

       The investigation was carried out on the basis of clinical sanatorium “Ukraine” (Yalta, Crimea) and department of laboratory studies of state educational, scientific and medical complex of clinic state institution “Crimea state medical university named after S. I. Georgievsky”. We formed 4 group of examined patients:1st group – 15 male patients with hypertension stage II, the mean age was 52±6,24 years, 2nd group - 15 female patients with hypertension stage II, the mean age was 51±6,15 year; 2 control group: 1st – 15 healthy young people, the mean age was 24±3,11; 2nd – 14 almost healthy men without arterial hypertension and CHD symptoms, the mean age – 51±5,48 years.

      Melatonin was measured in urine, collected in night time(from 21.00 to 6.00)

   In this way, the results of conducted investigation evidence that:

   1. The decrease of adaptive possibility in male patients having hypertension accompanied by low nocturnal excretion of melatonin metabolite (6 - 6-hydroxymelatoninsulphate (6–HMS))(p<,005) in comparison with control group. The female patients have more significant differences(p<0,001). After melatonin containing preparation using the difference of 6-HMS indexes in control and experimental group has leveled.

  2 . In spite of difference of indexes of 6-HMS excretion in men and women the adaptive potential of cardiovascular system in both groups has improved (on 16,35% in men and on 16,07% in women) and remained optimal after discontinuation of medication in 84% of patients.

In such a way after the receiving of melatonin drug course adaptation potential in males with hypertonic disease was equal to adequate functional possibilities of cardiovascular system (average adaptation), in females potential level changed from insufficient to intense level of adaptation. ). Simultaneously with decrease of arterial pressure patients felt better, up to normalization of “sleep-wake” processes and its circadian regulation with arterial pressure. Melatonin excretion in women is lower, this may be connected with endogenous melatonin production inhibition because of hyperprolactineemia. In such a way we may say that melatonin drugs prescribing patients with chronic hypertonic disease are very important because potential level changed from insufficient to intense level of adaptation.