Biological sciences / 9. Biochemistry and biophysics

                                  Bezrukaviy D.V., Rossikhin V.V.

National Technical University "Kharkiv Polytechnic Institute", Kharkiv city

ASSESSMENT OF THE ANTIOXIDIC ACTIVITY LEVEL OF BIOLOGICAL ACTIVE COMPOUNDS APPLYING ELECTROCHEMICAL METHODS

There exists a method that relates to the field of pharmaceutical chemistry and concerns the methods for quantitative determination of biologically active substances, in particular the total content of flavonoids –the substances with apparent antioxidant properties. The essence is: the transfer of substances from a sample (plant material) into a solution having the following voltammetric value, which is carried out using an indicator glass-carbon electrode with a saturated chloride silver electrode on the background of 0.1 mol/l of the phosphate buffer (pH 6.86) with the following recording of the anode peaks at a direct current form of the scan potential at the speed of 0.04 V/s. The concentration of the total content of flavonoids in the plant material is determined by the volume of the anode peak of the oxidation of substances at the range of potentials from +0.1 to +0.5V in a relatively saturated chlorine silver electrode. The area of ​​the determined content of the total amount of flavonoids ranges from 1õ10-5g/ml to 1õ10-4 g/ml.

Also there exists a well-known method that can be used in the food, cosmetic, pharmaceutical industries, as well as in medicine and forensic science. The proposed method allows measuring of the activity of antioxidants in relation to the most hazardous OH-radicals for the organism. In the process of recovering the substance on the electrode in the solution of the background electrolyte, a model reaction generating OH radicals is used, and the registration of the cathode waves of the recovery of the substance leads at the range of potentials -1.2 +- 1.9 V in a relatively saturated chlorine silver electrode comparison. In the indicated interval a peak appears, presumably, of OH-radicals, which decreases in proportion to the amount of added antioxidant. The activity of antioxidants is determined by the relative reduction of this peak.

The effect of the determination of the oxidant/antioxidant activity of the substances uses a method comprising the preparation of an initial solution with a mediator system containing both an oxidized and renovated form of a reagent and an evaluation of the oxidant/antioxidant activity on the grounds of the electrochemical parameters of the extract of the analyzed substance injected into the initial solution, and is characterized by the fact that the initial solution is divided into two volumes interconnected through a semipermeable membrane, and the extract of the test substance is injected into one of the volumes of the initial  solution and constant electromotive force is used as the electrochemical evaluation parameters of oxidant/antioxidant value in the measuring system.

Using this method allows increasing the accuracy and reliability of the information received.

There is an amperîmetric method that relates to the field of pharmacology and pharmacy, and can be used to evaluate the antioxidant activity (AOA) of various multicomponent mixtures without prior separation. The method involves the preparation of samples of the analyzed and standard substances, their electrochemical oxidation in the amperometric detector cell, the amplification of electrical signals for their registration, and the calculation of AOA from the proposed mathematical dependence. The method allows estimating the total antioxidant activity with high accuracy and reproductive performance and using simple and available equipment.

There is a new approach to the estimation of integral antioxidant capacity with the help of electrogenerated titrants. The antioxidant effect of 78 kinds of plants was investigated. For the quantitative assessment of antioxidant capacity, the proposed characteristic was implemented which was bromine antioxidant capacity (AOC), expressed in units of amount of electricity (coils), spent on titration of 100g (100 ml) of the preparation electro-generated by bromine. The relationship between the integral antioxidant capacity of food products, medicinal plant material and the content of individual groups of biologically active compounds was established: the sum of flavonoids, tocopherols and substances of a restorative nature.

It should be noted that not only one method for assessing the antioxidant activity of compounds exists, moreover it is quite complicated to compare the results obtained by different methods. In view of this it may be explained by the variety of radical processes occurring in nature.

However, in our opinion, the most appropriate method should be considered, in which the wave of electrolytic reduction O2 is used as a standard. Implementing the model reaction of the electrolytic reduction process O2, which follows the mechanism, similar to the restoration of oxygen in cells of the human body and animal, plant tissues and is the main oxidation process on all objects of artificial and natural origin, which makes this method more appealing.

In order to determine the total amount of antioxidants in the investigated object, a scalar is constructed which is relative to the change of the electrolytic reduction current O: from the concentration of ascorbic acid in the solution. Further out of this dependence on the value the relative change in the current in the presence of the object under study the total amount of antioxidants converted to the concentration of ascorbic acid is determined. This unified method also solves a number of problems associated with the absence of standard antioxidant samples and a standardized total antioxidant activity.